{"id":16473,"date":"2020-12-21T07:50:57","date_gmt":"2020-12-21T07:50:57","guid":{"rendered":"https:\/\/www.wholecelium.com\/?p=16473"},"modified":"2023-11-02T16:01:35","modified_gmt":"2023-11-02T15:01:35","slug":"vedci-vyrabeji-nehalucinogenni-ibogain","status":"publish","type":"post","link":"https:\/\/www.wholecelium.com\/cs\/blog\/scientists-make-non-hallucinogenic-ibogaine\/","title":{"rendered":"V\u011bdci vyrobili nehalucinogenn\u00ed ibogain"},"content":{"rendered":"<\/p>\n<\/p>\n<\/p>\n\n\n<\/p>\n<p><strong>Ta droga Darkstar? Jmenuje se ibogain.<\/strong><\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Naz\u00fdv\u00e1 se <strong>\"proti drog\u00e1m\"<\/strong> v\u011bdci i u\u017eivateli, se ibogain dostal na tituln\u00ed str\u00e1nky novin d\u00edky sv\u00fdm 99% \u00fasp\u011bch\u016fm v odvykac\u00edch programech. Mo\u017en\u00e1 jste o n\u011bm sly\u0161eli, mo\u017en\u00e1 ne. Koneckonc\u016f, u\u017e\u00edv\u00e1n\u00ed ibogainu je leg\u00e1ln\u00ed <em>pouze<\/em> na mexick\u00fdch klinik\u00e1ch a na n\u011bkolika dal\u0161\u00edch m\u00edstech, nap\u0159\u00edklad v Ji\u017en\u00ed Africe, Braz\u00edlii a na Nov\u00e9m Z\u00e9landu. Odvykac\u00ed l\u00e9\u010dba ibogainem je pom\u011brn\u011b drah\u00e1 - stoj\u00ed od <strong>$5,000 a\u017e $10,000 dolar\u016f<\/strong> pokud je u\u017e\u00edv\u00e1n s licencovan\u00fdm odborn\u00edkem - co\u017e je jedin\u00fd zp\u016fsob, jak by m\u011bl b\u00fdt u\u017e\u00edv\u00e1n. <em>(v\u00edce o tom pozd\u011bji).<\/em><\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Pokud je ibogain tak zatracen\u011b \u00fa\u010dinn\u00fd a siln\u00fd pro odvyk\u00e1n\u00ed drog, pro\u010d je v USA a dal\u0161\u00edch zem\u00edch, kter\u00e9 se zab\u00fdvaj\u00ed drogami, st\u00e1le neleg\u00e1ln\u00ed?<strong> <a href=\"https:\/\/www.drugabuse.gov\/drug-topics\/opioids\/opioid-overdose-crisis\" target=\"_blank\" rel=\"noreferrer noopener\">opioidov\u00e1 krize<\/a><\/strong>? Jednoduch\u00fd d\u016fvod: ibogain je halucinogenn\u00ed. To je d\u016fvod, pro\u010d je v USA tato droga za\u0159azena do seznamu 1 kontrolovan\u00fdch l\u00e1tek, tedy drog <em>\"bez l\u00e9ka\u0159sk\u00e9 hodnoty\"<\/em>. Nebo se to alespo\u0148 \u0159\u00edk\u00e1...<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Ale co kdyby v\u011bdci mohli <strong>vyjmout halucinogenn\u00ed \u010d\u00e1sti<\/strong> ibogainu, tak\u017ee z\u016fst\u00e1v\u00e1 pouze jeho potenci\u00e1l pro drogovou rehabilitaci? Bude <em>\"proti drog\u00e1m\"<\/em> kone\u010dn\u011b dekriminalizov\u00e1ny ve St\u00e1tech?&nbsp;<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Poj\u010fme to zjistit!<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<h2 class=\"wp-block-heading\" id=\"h-artificial-ibogaine\"><em> Um\u011bl\u00fd ibogain<\/em><\/h2>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Ibogain poch\u00e1z\u00ed z ko\u0159en\u016f rostliny zvan\u00e9 <strong>Tabernanthe iboga<\/strong>, kter\u00fd m\u00e1 halucinogenn\u00ed \u00fa\u010dinky. Jako psychedelick\u00e1 droga se v\u0161ak ibogain pou\u017e\u00edv\u00e1 jen z\u0159\u00eddka pro z\u00e1bavu, ale mimo jin\u00e9 jako solidn\u00ed zp\u016fsob l\u00e9\u010dby z\u00e1vislosti na opi\u00e1tech a alkoholu.<\/p>\n<p>\n\n\n<\/p>\n\n\n<figure class=\"wp-block-image size-full is-resized\"><img fetchpriority=\"high\" decoding=\"async\" width=\"740\" height=\"445\" src=\"https:\/\/www.wholecelium.com\/wp-content\/uploads\/Tabernanthe_iboga_bark_pieces.jpg\" alt=\"k\u016fra ibogainu s perem pro orientaci velikosti\" class=\"wp-image-159738\" style=\"width:841px\" srcset=\"https:\/\/www.wholecelium.com\/wp-content\/uploads\/Tabernanthe_iboga_bark_pieces.jpg 740w, https:\/\/www.wholecelium.com\/wp-content\/uploads\/Tabernanthe_iboga_bark_pieces-300x180.jpg 300w, https:\/\/www.wholecelium.com\/wp-content\/uploads\/Tabernanthe_iboga_bark_pieces-18x12.jpg 18w, https:\/\/www.wholecelium.com\/wp-content\/uploads\/Tabernanthe_iboga_bark_pieces-600x361.jpg 600w\" sizes=\"(max-width: 740px) 100vw, 740px\" \/><figcaption class=\"wp-element-caption\"><em><mark style=\"background-color:rgba(0, 0, 0, 0)\" class=\"has-inline-color has-cyan-bluish-gray-color\">K\u016fra z Tabernanthe iboga (zn\u00e1m\u00e1 tak\u00e9 jako \"prav\u00fd ibogain\"). via Wikipedia<\/mark><\/em><\/figcaption><\/figure>\n\n\n<\/p>\n\n\n<\/p>\n<p>Stejn\u011b jako u jin\u00fdch psychedelick\u00fdch l\u00e1tek jsou \u00fa\u010dinky ibogainu dlouhodob\u00e9. V\u011bdci to d\u00e1vaj\u00ed do souvislosti se schopnost\u00ed ibogainu <strong><em>\"p\u0159epojit\"<\/em> mozkov\u00e9 vzorce<\/strong> se z\u00e1vislost\u00ed... ale to se m\u016f\u017ee st\u00e1t pouze uprost\u0159ed roku. <em>\"re\u017eim paral\u00fdzy\"<\/em>.<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Na\u0161t\u011bst\u00ed pro ty, kter\u00fdm by l\u00e9\u010dba ibogainem prosp\u011bla, bude mo\u017en\u00e1 brzy mo\u017en\u00e9 paral\u00fdzu p\u0159esko\u010dit. V\u011bdci z v\u00fdzkumn\u00e9ho \u00fastavu pro l\u00e9\u010dbu ibogainem p\u0159ipravili verzi ibogainu bez tripu. <strong>Katedra chemie UC Davis<\/strong>, jak bylo zve\u0159ejn\u011bno v \u010dasopise Nature 9. prosince.<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p><strong>David Olson<\/strong>, odborn\u00fd asistent chemie na Kalifornsk\u00e9 univerzit\u011b v Davisu a hlavn\u00ed autor \u010dl\u00e1nku, \u0159ekl:<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p><em>\"Psychedelika jsou jedny z nejsiln\u011bj\u0161\u00edch drog, kter\u00e9 zn\u00e1me a kter\u00e9 ovliv\u0148uj\u00ed mozek. Je neuv\u011b\u0159iteln\u00e9, jak m\u00e1lo o nich v\u00edme.\"<\/em><\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Olsonova laborato\u0159 na Kalifornsk\u00e9 univerzit\u011b v Davisu, kter\u00e1 m\u00e1 jako jedna z m\u00e1la licenci na nakl\u00e1d\u00e1n\u00ed s l\u00e1tkami za\u0159azen\u00fdmi do seznamu 1, vytvo\u0159ila<strong> analogov\u00fd<\/strong> <em>(nebo bl\u00edzk\u00e1 kopie)<\/em> ibogainu, kter\u00fd si zachoval sv\u00e9 \u00fa\u010dinky proti z\u00e1vislosti a z\u00e1rove\u0148 odstranil sv\u00e9 halucinogenn\u00ed \u00fa\u010dinky.&nbsp;<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Po z\u00e1m\u011bn\u011b \u010d\u00e1st\u00ed molekuly ibogainu za \u0159adu podobn\u00fdch slou\u010denin. <em>(jak\u00e9si Frankensteinovo monstrum v podob\u011b molekuly).<\/em>, Olsonova laborato\u0159 skon\u010dila s novou um\u011blou molekulou, tzv. <strong>TBG<\/strong>, nebo<strong> tabernanthalog<\/strong>.<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<h2 class=\"wp-block-heading\" id=\"h-less-toxic-than-ibogaine\"> <em>M\u00e9n\u011b toxick\u00fd ne\u017e ibogain? <\/em><\/h2>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Na tomto m\u00edst\u011b v\u00e1m mus\u00edme \u0159\u00edci, \u017ee ibogain m\u00e1 dal\u0161\u00ed vedlej\u0161\u00ed \u00fa\u010dinky, kter\u00e9 se poj\u00ed s jeho potenci\u00e1lem proti z\u00e1vislosti. Za prv\u00e9, ibogain m\u016f\u017ee vyvolat srde\u010dn\u00ed z\u00e1chvaty. Za druh\u00e9 je tak\u00e9 vysoce toxick\u00fd - zp\u016fsobuje mnoho \u00famrt\u00ed v d\u016fsledku nedostate\u010dn\u00e9ho nebo nespr\u00e1vn\u00e9ho dohledu.<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Studie UC Davis vyzkou\u0161ela TBG na bun\u011b\u010dn\u00fdch kultur\u00e1ch a zeb\u0159i\u010dk\u00e1ch a zjistila, \u017ee TBG je daleko \u00fa\u010dinn\u011bj\u0161\u00ed ne\u017e TBG. <strong>m\u00e9n\u011b toxick\u00e9<\/strong> ne\u017e ibogain. Uff!&nbsp;<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Testovali tak\u00e9 na nervov\u00fdch bu\u0148k\u00e1ch potkan\u016f, kde TBG <strong>urychlil r\u016fst<\/strong> nov\u00fdch dendrit\u016f <em>(pobo\u010dky)<\/em> - co\u017e je vlastn\u011b dost podobn\u00e9 tomu, jak LSD a DMT spou\u0161t\u011bj\u00ed nov\u00e9 mozkov\u00e9 bu\u0148ky.&nbsp;<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<h2 class=\"wp-block-heading\" id=\"h-no-more-opiate-relapses\"> <em>U\u017e \u017e\u00e1dn\u00e9 relapsy opi\u00e1t\u016f  <\/em><\/h2>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Kdy\u017e u\u017e mluv\u00edme o krys\u00e1ch, TBG prok\u00e1zal na modelech hlodavc\u016f \u0161\u00edlen\u00fd potenci\u00e1l pro potla\u010den\u00ed z\u00e1vislosti a deprese. Nap\u0159\u00edklad my\u0161i, kter\u00e9 byly vycvi\u010deny k pit\u00ed alkoholu. <strong>se stal <em>\"st\u0159\u00edzliv\u00fd\"<\/em><\/strong> ji\u017e po jedn\u00e9 d\u00e1vce TBG.&nbsp;<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Ostatn\u00ed my\u0161i byly nau\u010deny stisknout p\u00e1\u010dku pro <strong>d\u00e1vka heroinu<\/strong> kdykoli se rozsv\u00edt\u00ed sv\u011btlo s t\u00f3nem. Po odstran\u011bn\u00ed opi\u00e1tu se u potkan\u016f objevily abstinen\u010dn\u00ed p\u0159\u00edznaky - co\u017e je p\u0159im\u011blo znovu stisknout p\u00e1ku. Ale po TBG se u potkan\u016f objevil relaps. <strong>trvalo d\u00e9le, ne\u017e se vyno\u0159il<\/strong>, pokud v\u016fbec!<\/p>\n<p>\n\n\n<\/p>\n\n\n<figure class=\"wp-block-image size-full is-resized\"><img decoding=\"async\" width=\"709\" height=\"399\" src=\"https:\/\/www.wholecelium.com\/wp-content\/uploads\/hallucination-trick-of-the-eye-picture.jpeg\" alt=\"psychedelick\u00e1 barevn\u00e1 spir\u00e1la\" class=\"wp-image-159743\" style=\"width:841px\" srcset=\"https:\/\/www.wholecelium.com\/wp-content\/uploads\/hallucination-trick-of-the-eye-picture.jpeg 709w, https:\/\/www.wholecelium.com\/wp-content\/uploads\/hallucination-trick-of-the-eye-picture-300x169.jpeg 300w, https:\/\/www.wholecelium.com\/wp-content\/uploads\/hallucination-trick-of-the-eye-picture-18x10.jpeg 18w, https:\/\/www.wholecelium.com\/wp-content\/uploads\/hallucination-trick-of-the-eye-picture-600x338.jpeg 600w\" sizes=\"(max-width: 709px) 100vw, 709px\" \/><\/figure>\n\n\n<\/p>\n\n\n<p><\/p>\n\n\n<\/p>\n\n\n<h2 class=\"wp-block-heading has-pale-cyan-blue-color has-text-color\" id=\"h-a-drug-that-people-keep-in-their-medicine-cabinet\"><em> \"Droga, kterou maj\u00ed lid\u00e9 v l\u00e9k\u00e1rni\u010dce\" <\/em><\/h2>\n\n\n<\/p>\n\n\n<\/p>\n<p>Skute\u010dn\u00fd ibogain nen\u00ed rozpustn\u00fd ve vod\u011b a vy\u017eaduje mnoho f\u00e1z\u00ed, jen aby se dostal do va\u0161eho syst\u00e9mu. Na druhou stranu TBG, <strong>v\u0161echny tyto kroky p\u0159esko\u010d\u00ed<\/strong> pro t\u00e9m\u011b\u0159 okam\u017eit\u00fd \u00fa\u010dinek. Je to z\u00e1sadn\u00ed v\u011bc, kterou je t\u0159eba zv\u00e1\u017eit, pokud se psychedelick\u00e9 l\u00e9ky skute\u010dn\u011b cht\u011bj\u00ed st\u00e1t alternativou k velk\u00e9 farmacii. Jak \u0159ekl Olson:<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p><em>\"Pot\u0159ebujeme l\u00e9k, kter\u00fd by lid\u00e9 mohli m\u00edt ve sv\u00e9 l\u00e9k\u00e1rni\u010dce, a toto je v\u00fdznamn\u00fd krok t\u00edmto sm\u011brem.\"<\/em><\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Nyn\u00ed v\u00edme, \u017ee TBG m\u016f\u017ee dos\u00e1hnout stejn\u00fdch c\u00edl\u016f jako ibogain, pokud jde o p\u0159epojov\u00e1n\u00ed z\u00e1vislost\u00ed. M\u016f\u017ee v\u0161ak TBG l\u00e9\u010dit i \u0159adu dal\u0161\u00edch stav\u016f, jako nap\u0159. <strong>deprese<\/strong>, <strong>\u00fazkost<\/strong>a <strong>PTSD<\/strong>?&nbsp;<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Pro\u010d ne, \u0159\u00edk\u00e1 Olson:<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p><em>\"Dosud jsme se zam\u011b\u0159ovali na l\u00e9\u010dbu jednoho psychiatrick\u00e9ho onemocn\u011bn\u00ed najednou, ale v\u00edme, \u017ee se tato onemocn\u011bn\u00ed p\u0159ekr\u00fdvaj\u00ed. Mohlo by b\u00fdt mo\u017en\u00e9 l\u00e9\u010dit v\u00edce nemoc\u00ed stejn\u00fdm l\u00e9kem.\"<\/em><\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Psychedelick\u00e9 terapie se t\u011b\u0161\u00ed velk\u00e9 oblib\u011b.<strong> <a href=\"https:\/\/www.wholecelium.com\/cs\/articles\/politicky\/psychedelika-vlna-se-blizi\/\" target=\"_blank\" rel=\"noreferrer noopener\">comeback<\/a><\/strong>, verze hippie revoluce z 60. let 21. stolet\u00ed. Na rozd\u00edl od na\u0161ich p\u0159edch\u016fdc\u016f v\u0161ak nem\u016f\u017eeme br\u00e1t pacienty na v\u00fdlety po jednom. \u017dere to drahocenn\u00fd \u010das a pen\u00edze - nemluv\u011b o p\u0159\u00edsn\u00e9m l\u00e9ka\u0159sk\u00e9m dohledu. Nen\u00ed to sch\u016fdn\u00e1 varianta, pokud chceme dos\u00e1hnout skute\u010dn\u00fdch zm\u011bn v l\u00e9\u010db\u011b obrovsk\u00e9ho mno\u017estv\u00ed vy\u010derp\u00e1vaj\u00edc\u00edch onemocn\u011bn\u00ed.<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<h2 class=\"wp-block-heading\" id=\"h-strictly-for-healing\"><em>P\u0159\u00edsn\u011b pro l\u00e9\u010den\u00ed<\/em><\/h2>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>P\u0159esto\u017ee je ibogain pova\u017eov\u00e1n za \"psychedelickou drogu\", nejedn\u00e1 se o rekrea\u010dn\u00ed drogu. Je pravda, \u017ee n\u011bkter\u00e1 psychedelika, jako je psilocybin, lze u\u017e\u00edvat jak terapeuticky, tak rekrea\u010dn\u011b, ale ibogain pat\u0159\u00ed do kategorie \"v\u00fdhradn\u011b l\u00e9\u010debn\u00fdch\". Jak v\u0161ak bude pokra\u010dovat v\u00fdzkum prosp\u011b\u0161nosti v\u0161ech druh\u016f psychedelik, jejich jednotliv\u00e9 pokroky si budou vz\u00e1jemn\u011b pom\u00e1hat v \u00fasil\u00ed o legalizaci a zviditeln\u011bn\u00ed. <\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Co si o tom mysl\u00edte? Bude ibogain dal\u0161\u00ed drogou, kter\u00e1 bude <strong>dekriminalizace<\/strong>  nyn\u00ed, kdy\u017e m\u00e1 variantu bez v\u00fdletu?<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>Pod\u011blte se o sv\u00e9 n\u00e1zory n\u00ed\u017ee!<\/p>\n<p>\n\n\n<\/p>\n\n\n<\/p>\n<p>P.S. Pro hlub\u0161\u00ed a \u00fapln\u011bj\u0161\u00ed ponor do problematiky ibogainu <em>(a jeho \u0161\u00edlen\u00e1 historie)<\/em>, pod\u00edvejte se na tento&nbsp;<a href=\"https:\/\/www.wholecelium.com\/cs\/blog\/jak-ibogain-meni-zivoty\/\" target=\"_blank\" rel=\"noopener\"><b>\u010dl\u00e1nek<\/b><\/a><strong>. <\/strong><\/p>\n<p>\n\n\n<\/p>","protected":false},"excerpt":{"rendered":"<p>Not all psychedelic compounds are the same. Most recreational psychedelics \u2014 such as psilocybin, LSD, and MDMA \u2014 trigger a cacophony of colours and sensations in a zip-zap trip to Wonderland. One substance, however, does the exact opposite&#8230; paralyzing you in a waking dream, static and unmoving.\u00a0<\/p>","protected":false},"author":1,"featured_media":16474,"comment_status":"open","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[68],"tags":[],"topics":[],"class_list":["post-16473","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-science-and-studies"],"_links":{"self":[{"href":"https:\/\/www.wholecelium.com\/cs\/wp-json\/wp\/v2\/posts\/16473","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/www.wholecelium.com\/cs\/wp-json\/wp\/v2\/posts"}],"about":[{"href":"https:\/\/www.wholecelium.com\/cs\/wp-json\/wp\/v2\/types\/post"}],"author":[{"embeddable":true,"href":"https:\/\/www.wholecelium.com\/cs\/wp-json\/wp\/v2\/users\/1"}],"replies":[{"embeddable":true,"href":"https:\/\/www.wholecelium.com\/cs\/wp-json\/wp\/v2\/comments?post=16473"}],"version-history":[{"count":6,"href":"https:\/\/www.wholecelium.com\/cs\/wp-json\/wp\/v2\/posts\/16473\/revisions"}],"predecessor-version":[{"id":159745,"href":"https:\/\/www.wholecelium.com\/cs\/wp-json\/wp\/v2\/posts\/16473\/revisions\/159745"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/www.wholecelium.com\/cs\/wp-json\/wp\/v2\/media\/16474"}],"wp:attachment":[{"href":"https:\/\/www.wholecelium.com\/cs\/wp-json\/wp\/v2\/media?parent=16473"}],"wp:term":[{"taxonomy":"category","embeddable":true,"href":"https:\/\/www.wholecelium.com\/cs\/wp-json\/wp\/v2\/categories?post=16473"},{"taxonomy":"post_tag","embeddable":true,"href":"https:\/\/www.wholecelium.com\/cs\/wp-json\/wp\/v2\/tags?post=16473"},{"taxonomy":"topics","embeddable":true,"href":"https:\/\/www.wholecelium.com\/cs\/wp-json\/wp\/v2\/topics?post=16473"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}